LONG-TERM (AT LEAST 24 MONTHS)

TOXICITY

PURPOSE:

A broad screen for toxicity that will define effects, establish the NOEL, and determine carcinogenicity

ANIMALS:

Rodents-50/sex/group with increases for sacrifices planned before the end of the test.

Dogs-8/sex/group

DOSAGE:

At least three plus control.

Lowest dose should not show toxicity.

At least 50% of the animals should survive for 24 months.

The highest dose is usually the highest amount that can be administered without reducing the life span of the animals unless that dose exceeds 5% of the diet.

OBSERVATIONS:

Daily observations similar to sub-chronic studies.

Histopathology to include:

Adrenal

Peripheral Nerve

Aorta

Pituitary

Bone

Prostate

Bone Marrow

Rectum

Brain (3+Levels)

Rep. Lymph Nodes

Caecum

Salivary Glands

Colon

Seminal Vesicle

Corpus & Cervis Uteri

Skeletal Muscle

Duodenum

Smooth Muscle

Esophagus

SpinalCord (2+Levels)

Eyes

Spleen

Gall Bladder

Sternum

Heart

Stomach

Ileum

Testes

Jejunum

Thymus

Kidneys

Thyroid (Parathyroid)

Liver

Trachea

Lungs

Urinary Bladder

Mammery Glands

All tissues showing abnormality

Ovaries

 

Pancreas